PreclinicalHealing & RecoveryWADA-banned

TB-500

A synthetic fragment marketed as thymosin beta-4 · "TB4 lite"

Overview

TB-500 is a synthetic peptide sold for recovery from injury, inspired by a fragment of the natural protein thymosin beta-4. It is not an approved medicine anywhere, evidence in humans is essentially absent, and it is banned at all times in tested sport by WADA.

01 What is TB-500?

In plain English.

TB-500 is a lab-made peptide marketed as a recovery aid. Its name is a marketing label, not a scientific one: it refers to a shortened, synthetic sequence inspired by thymosin beta-4 (TB-4), a 43-amino-acid protein the body produces naturally, particularly at sites of injury. The vials sold to bodybuilders and gym-goers are not the same molecule as the full TB-4 used in clinical research, although vendors often blur the two.

⏱ Half-life
~Hours (est. animal)
☉ Route
Subcutaneous / IM
⚖ Evidence
Preclinical
📚 Studies
5 referenced

This distinction matters: when you read about TB-4 healing corneas or repairing heart tissue in animal studies, that work was done with the full 43-residue protein (or its drug form, RGN-259), not the fragment sold online as "TB-500". Treat the two as related-but-different, and assume any TB-4 evidence transfers to TB-500 only loosely.

02 How it works

The simple version, then the science.

In animals, thymosin beta-4 appears to help injured tissue rebuild itself: it promotes new blood-vessel formation (angiogenesis), recruits cells that migrate into wounds, and dampens inflammation. The marketed TB-500 fragment is claimed to recapitulate these actions, on the basis that it includes the short "actin-binding" region thought to do much of the work.

Go deeper · the proposed mechanism

TB-4 is the most abundant member of the beta-thymosin family and binds G-actin, sequestering monomers and regulating cytoskeletal dynamics during cell migration. In rodent models it has been reported to upregulate VEGF and integrin-linked kinase (ILK) signalling, stimulate endothelial cell migration, and modulate inflammatory cytokines. These mechanisms are described for the full protein; whether the truncated TB-500 fragment produces the same downstream effects in humans is not established.

03 What it's used for

Each use graded by how strong the evidence actually is.

  • Preclinical
    Soft-tissue & wound healingRepeated rodent studies on dermal, corneal and cardiac wounds, using full TB-4, not the marketed fragment. No controlled human trials of TB-500 itself.
  • Preclinical
    Cardiac repair after injuryA 2004 Nature paper showed TB-4 protected mouse heart cells after infarct. Promising preclinical signal; not yet translated to humans.
  • Anecdotal
    Tendon, ligament & muscle recovery in athletesPopular in performance circles, often stacked with BPC-157. Supported only by self-reports.
  • Anecdotal
    Hair regrowthFrequently claimed online. No controlled human data.
Banned in tested sport. Thymosin beta-4 and its fragments are prohibited at all times by WADA under S2 (Peptide Hormones, Growth Factors, Related Substances and Mimetics). No use of TB-500 is supported by approved human clinical trials.

04 What the evidence says

Most of the science people cite under "TB-500" is actually evidence for the full thymosin beta-4 protein, and even that is overwhelmingly preclinical. RegeneRx's drug candidate RGN-259, an ophthalmic formulation of full TB-4, has progressed through Phase 2/3 trials for dry eye and corneal injury, with mixed results across primary endpoints. There are essentially no controlled human trials of the shortened "TB-500" fragment that's sold online. Animal results for wound healing and cardiac repair are real and reproducible in the literature, but the gap between a mouse and a human is wide, and the gap between full TB-4 and a marketing-named fragment widens it further. In short: an interesting preclinical signal for TB-4, very weak read-across to TB-500, and no proven human benefit.

05 Dosing & administration

Reported in the literature, information not advice.

Because there is no approved human protocol, no safe or effective dose has been established. Online communities describe milligram-range subcutaneous injections, often weekly, but these regimens are not backed by clinical evidence and the purity of research-grade vials is not regulated. A qualified clinician should be consulted before considering any peptide.

06 Side effects & safety

Long-term safety in humans is unknown, there are no large clinical trials of TB-500. Short-term reports from users include injection-site reactions and occasional lethargy. A specific theoretical concern is that TB-4 promotes angiogenesis (blood-vessel growth), which could in principle accelerate the growth of existing tumours; this has not been demonstrated clinically but is a reasonable reason for caution in anyone with cancer or a cancer history. Products sold as "TB-500" are unregulated research chemicals, contamination, mislabelling and dose-by-dose variation are real risks. People who are pregnant, breastfeeding, immunocompromised, or taking other medicines should be especially cautious.

WADA-banned · not approved anywhere. TB-500 is on the WADA Prohibited List at all times under S2. Sold legally only as a research chemical, not for human consumption.

07 Where to buy (research use only)

Vetted on quality and transparency, not an endorsement to use.

Helix Research Labs4.6
Research-use-only peptides with publicly available certificates of analysis.
HPLC & MS verifiedPublished COAsResearch use only
View ↗
Apex Compounds4.3
Competitive pricing across a broad range of research compounds.
Third-party testedResearch use only
View ↗
Vanta Bio4.5
Specialist supplier with independent lab testing on every batch.
Independent lab testingResearch use only
View ↗
Disclosure: Pepwyse is not affiliated with these companies and does not earn any commission from these links; they are listed for reference only. These products are sold strictly for laboratory research use only and are not for human consumption.

09 Clinical studies & research

Primary sources. Read the science yourself.

Thymosin β4 activates integrin-linked kinase and promotes cardiac cell migration, survival and cardiac repair
Nature · 2004 Animal (mouse)
Landmark study showing full TB-4 protected mouse heart cells after infarct and improved cardiac function. The most-cited preclinical paper underlying TB-4 / TB-500 marketing claims. View on PubMed →
β-Thymosins
Annals of the New York Academy of Sciences · 2007 Review
Overview of the beta-thymosin family, biology, actin-binding role, and the rationale for therapeutic interest in TB-4. Useful for grounding the science behind the marketing. View on PubMed →
Thymosin beta-4: a novel corneal wound healing and anti-inflammatory agent
Clinical Ophthalmology · 2007 Review / preclinical
Summarises the preclinical case for TB-4 in corneal wound healing, the basis for RegeneRx's drug candidate RGN-259. View on PubMed →
Thymosin β4 and the eye: the journey from bench to bedside
Expert Opinion on Biological Therapy · 2018 Review
Tracks TB-4 (full protein, as RGN-259) through Phase 2/3 ophthalmic trials for dry eye and corneal injury. The clearest summary of the actual human clinical record, none of it concerns the marketed "TB-500" fragment. View on PubMed →
Thymosin β4 Promotes Dermal Healing
Vitamins and Hormones · 2016 Review · preclinical
Synthesises rodent dermal-wound studies on TB-4. Reproducible preclinical signal; not a human trial. View on PubMed →

10 Frequently asked questions

Is TB-500 the same thing as thymosin beta-4?
No, and this matters. Thymosin beta-4 (TB-4) is a 43-amino-acid protein the body produces naturally. "TB-500" is a marketing name for a shorter synthetic fragment inspired by TB-4. The full TB-4 protein has been studied in human clinical trials as the drug candidate RGN-259; the shortened TB-500 fragment sold online has not.
Is TB-500 banned in sport?
Yes. Thymosin beta-4 and its fragments are prohibited at all times under the WADA Prohibited List, S2 (Peptide Hormones, Growth Factors, Related Substances and Mimetics). It is also banned by equine anti-doping bodies, multiple racehorse positives have been reported.
Is TB-500 approved by any regulator?
No. TB-500 is not approved as a medicine in the UK, US, EU, Australia or Canada. It is sold only as a research chemical, not for human consumption.
Does TB-500 actually heal injuries?
In animals, the parent protein TB-4 shows reproducible wound-healing effects. In humans, the evidence is essentially absent for the shortened TB-500 fragment that is actually sold. Honest answer: unproven.
Is TB-500 safe?
Its safety profile in humans is unknown. There are no large human trials. Theoretical concerns include the angiogenic effects of TB-4 in anyone with cancer history. Products sold online are unregulated and quality varies.
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